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Inhibition of human DHODH
Assay data:21 Active, 8 Activity ≤ 1 µM, 21 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Primary qHTS for Inhibitors of ATXN expression
Assay data:2593 Active, 3 Activity ≤ 1 nM, 2671 Activity ≤ 1 µM, 361713 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Cytochrome P450 Family 1 Subfamily A Member 2 (CYP1A2) small molecule antagonists: luciferase reporter qHTS assay
Assay data:2934 Active, 132 Activity ≤ 1 µM, 9667 Tested
Primary qHTS for Inhibitors of N-terminal methyltransferase 1 (NTMT1): MTaseGlo Assay
Assay data:1477 Active, 244 Activity ≤ 1 µM, 58936 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Validation qHTS assay for inhibitors of Activation Induced Cytidine Deaminase (AID): AID signal
Assay data:18 Active, 39 Activity ≤ 1 µM, 1279 Tested
Human pregnane X receptor (PXR) activation by small molecules, qHTS assay
Assay data:229 Active, 16 Activity ≤ 1 µM, 2454 Tested
Identifying Small Molecule Inhibitors of Pancreatic Cancer Stem Cells (Panc1, Spheroid)
Assay data:67 Active, 5 Activity ≤ 1 nM, 143 Activity ≤ 1 µM, 464 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same Project
qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line in the presence of 0.5 nM R1881
Assay data:1453 Active, 4 Activity ≤ 1 nM, 292 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS assay for measurement of the activity of small molecule inhibitors on Zika virus induced Caspase-3 activity in human iPSC derived neural progenitor cells (hNPCs)
Assay data:110 Active, 1 Activity ≤ 1 nM, 91 Activity ≤ 1 µM, 5704 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
qHTS assay to identify small molecule agonists of the constitutive androstane receptor (CAR) signaling pathway
Assay data:853 Active, 48 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS assay to identify small molecule antagonists of the constitutive androstane receptor (CAR) signaling pathway
Assay data:575 Active, 6 Activity ≤ 1 nM, 184 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway
Assay data:1034 Active, 2 Activity ≤ 1 nM, 491 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule agonists of the endoplasmic reticulum stress response signaling pathway - cell viability counter screen
Assay data:328 Active, 5 Activity ≤ 1 nM, 337 Activity ≤ 1 µM, 9315 Tested
qHTS profiling for inhibitors of Plasmodium falciparum (3D7) proliferation
Assay data:16 Activity ≤ 1 nM, 124 Activity ≤ 1 µM, 633 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same Project
qHTS assay to identify aromatase inhibitors
Assay data:905 Active, 3 Activity ≤ 1 nM, 352 Activity ≤ 1 µM, 10486 Tested
qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway - cell viability counter screen
Assay data:583 Active, 15 Activity ≤ 1 nM, 316 Activity ≤ 1 µM, 10486 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same Project
qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rev3 mutant cell line
Assay data:2493 Active, 2 Activity ≤ 1 nM, 413 Activity ≤ 1 µM, 10486 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT
Assay data:49946 Active, 2 Activity ≤ 1 nM, 3516 Activity ≤ 1 µM, 424035 Tested
Cell Proliferation Assay against the HBL1 Cell Line
Assay data:5 Activity ≤ 1 nM, 67 Activity ≤ 1 µM, 461 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same Project
DRUGMATRIX: CYP450, 1A2 enzyme inhibition (substrate: 3-Cyano-7-ethoxycoumarin)
Assay data:40 Active, 23 Activity ≤ 1 µM, 871 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
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