Strategies at the interface of drug discovery and development: early optimization of the solid state phase and preclinical toxicology formulation for potential drug candidates

J Med Chem. 2010 Aug 26;53(16):5897-905. doi: 10.1021/jm1002638.
No abstract available

MeSH terms

  • Animals
  • Chemistry, Pharmaceutical
  • Crystallization
  • Drug Compounding*
  • Drug Discovery / methods*
  • Drug Evaluation, Preclinical
  • Drug Stability
  • Humans
  • Pharmaceutical Preparations / chemistry*
  • Pharmaceutical Preparations / metabolism
  • Pharmacokinetics
  • Solubility
  • Toxicity Tests

Substances

  • Pharmaceutical Preparations