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Neuroprotective activity against transgenic Caenorhabditis elegans CL2355 assessed as A-beta aggregration-induced reversal of disrupted chemotaxis behaviour by measuring chemotaxis index at 1.5 uM treated for 72 hrs followed by compound washout and odorant addition for 1 hr
Assay data:2 Active, 2 Tested
SummaryCompounds, ActivePubMed Citation
Effect on locomotory activity in transgenic Caenorhabditis elegans CL2006 model of paralysis assessed as reduction in defective locomotion by measuring motor index at 0.1 to 10 uM by motor behaviour assay
Antihelminthic activity against Caenorhabditis elegans N2 assessed as reduction in worm motility measured after 2 days by binocular dissecting microscopy
Assay data:6 Tested
SummaryPubMed Citation
Nematicidal activity against Caenorhabditis elegans incubated for 18 hrs
Assay data:8 Tested
Anthelmintic activity against Ancylostoma ceylanicum isolated from infected Syrian hamster feces assessed as reduction in motility at 25 ug/ml measured on day 5
Assay data:1 Tested
Inhibition of GST-tagged Caenorhabditis elegans CRN-4 exonuclease activity expressed in Escherichia coli BL21 (DE3) pLysS preincubated for 10 mins followed by [gamma-32P]ATP labelled 11-nucleotide ssRNA substrate addition for 30 mins by PAGE based autoradiography
Assay data:2 Active, 9 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Nematocidal activity against Caenorhabditis elegans assessed as mortality
Nematicidal activity against Caenorhabditis elegans assessed as immobility
Assay data:19 Tested
Toxicity in L4-stage of Caenorhabditis elegans expressing dpy-18 assessed as embyronic lethality after 24 hrs by light microscopic analysis
Nematicidal activity against Caenorhabditis elegans after 2 days
Nematocidal activity against Haemonchus contortus Haecon 5 strain isolated from helminth-free Merino weaner sheep after 6 days by larval development assay
Assay data:4 Active, 7 Tested
Inhibition of huntingtin mutant in Caenorhabditis elegans ASH neuronal cell Huntington disease model assessed as cell viability
Assay data:29 Tested
Antinematodal activity against Caenorhabditis elegans after 24 hrs by microscopy
Assay data:9 Tested
Antinematodal activity against Caenorhabditis elegans after 16 to 24 hrs
Anthelmintic activity against Caenorhabditis elegans
Anthelmintic activity against mice, infected with parasite Nematospiroides dubius, at a dose of 125 (ppm in feed)
Assay data:47 Tested
Compound was evaluated for the biological activity by Caenorhabditis elegans motility assay.
Tested in vitro for the biological efficacy using Caenorhabditis elegans binding assay; no data.
Assay data:4 Tested
Summary
Anthelmintic activity against third stage larvae of Haemonchus contortus assessed as inhibition of larval development at 20 uM measured after 7 days by microscopic analysis
Assay data:7 Tested
Anthelmintic activity against third stage larvae of Haemonchus contortus assessed as inhibition of xL3 larval motility at 20 uM measured after 72 hrs
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