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Antileishmanial activity against Leishmania mexicana mexicana BEL21 after 48 hrs
Assay data:3 Tested
SummaryPubMed Citation
Antileishmanial activity against Leishmania mexicana mexicana MHOM/BZ/84/BEL46 promastigotes assessed as parasite LDH activity by three-fold serial dilution method
Assay data:24 Tested
qHTS Assay for Inhibitors of Leishmania Mexicana Pyruvate Kinase (LmPK): Summary
Assay data:3 Active, 3 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
Confirmation Assay for Inhibitors of Leishmania Mexicana Pyruvate Kinase (LmPK): for Probe SAR
Assay data:38 Active, 2 Activity ≤ 1 nM, 24 Activity ≤ 1 µM, 225 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS Validation Assay for Activators of Leishmania Mexicana Pyruvate Kinase
Assay data:21 Active, 5 Activity ≤ 1 µM, 1279 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS Validation Assay for Inhibitors of Leishmania Mexicana Pyruvate Kinase
Assay data:22 Active, 5 Activity ≤ 1 µM, 1279 Tested
qHTS Assay for Activators of Leishmania Mexicana Pyruvate Kinase (LmPK)
Assay data:16 Activity ≤ 1 µM, 293196 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS Assay for Inhibitors of Leishmania Mexicana Pyruvate Kinase (LmPK)
Assay data:1089 Active, 16 Activity ≤ 1 µM, 293196 Tested
Confirmation Assay for Inhibitors of Leishmania Mexicana Pyruvate Kinase (LmPK)
Assay data:58 Active, 1 Activity ≤ 1 µM, 150 Tested
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