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Antileishmanial activity against promastigote stage of Leishmania donovani MHOM/PE/84/LC26 incubated for 72 hrs by Neubauer haemocytometric chamber analysis
Assay data:1 Tested
SummaryPubMed Citation
Antileishmanial activity against amastigote stage of Leishmania donovani MHOM/ET/67/HU3 infected in po dosed BALB/c mouse assessed as reduction in parasitemia administered twice a day for 10 days
Antileishmanial activity against amastigote stage of Leishmania donovani MHOM/ET/67/HU3 infected in BALB/c mouse assessed as reduction in parasitemia at 25 mg/kg, po bid for 10 days
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed Citation
Antileishmanial activity against amastigote stage of Leishmania donovani MHOM/ET/67/HU3 infected in BALB/c mouse assessed as reduction in parasitemia at 50 mg/kg, ip bid for 5 days
Inhibition of chymotrypsin activity of proteasome beta5 subunit in Leishmania donovani amastigotes infected in human THP-1 cells incubated for 96 hrs by INMAC assay
Assay data:27 Active, 16 Activity ≤ 1 µM, 45 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Antiparasitic activity against amastigote stage Leishmania donovani MHOM/ET/67/L82 infected in CD-1 mouse peritoneal macrophage assessed as reduction in parasite burden incubated for 5 days by Giemsa staining based microscopy
Assay data:3 Tested
Antiprotozoal activity against Leishmania donovani
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Antileishmanial activity against Leishmania donovani MHOM/ET/67:LV82 amastigotes infected in BMDM cell measured after 48 hrs by luciferase assay
Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested
Antileishmanial activity against Leishmania donovani promastigotes assessed as parasite growth inhibition incubated for 72 hrs by Alamar blue assay
Assay data:4 Tested
Antileishmanial activity against Leishmania donovani infected in human THP-1 cells assessed as growth inhibition at 100 uM by intramacrophage assay
Assay data:20 Tested
Antileishmanial activity against Leishmania donovani infected in human THP-1 cells assessed as growth inhibition by intramacrophage assay
Assay data:26 Active, 8 Activity ≤ 1 µM, 108 Tested
Antileishmanial activity against Leishmania donovani axenic amastigotes assessed as growth inhibition by fluorescence intensity readout assay
Assay data:2 Active, 2 Tested
Antileishmanial activity against Leishmania donovani amastigotes assessed as parasite growth inhibition
Assay data:1 Active, 3 Tested
Antileishmanial activity against Leishmania donovani assessed as parasite growth inhibition
Antileishmanial activity against Leishmania donovani D10 promastigotes assessed as parasite growth inhibition incubated for 24 hrs by alamar blue staining based analysis
Induction of cell cycle arrest in Leishmania donovani MHOM/IN/80/Dd8 promastigotes assessed as increase in subG0/G1 phase at 50 uM incubated for 72 hrs by PI staining based flow cytometry
Induction of apoptosis in Leishmania donovani MHOM/IN/80/Dd8 promastigotes assessed as breakdown of nuclear DNA at 50 uM incubated for 72 hrs by agarose gel electrophoresis
Induction of apoptosis in Leishmania donovani MHOM/IN/80/Dd8 promastigotes assessed as ladder like DNA at 50 uM incubated for 72 hrs by agarose gel electrophoresis
Induction of apoptosis in Leishmania donovani MHOM/IN/80/Dd8 promastigotes assessed as decrease in cytochrome c level in mitochondria at 50 uM incubated upto 48 hrs by immunoblot analysis
Induction of apoptosis in Leishmania donovani MHOM/IN/80/Dd8 promastigotes assessed as increase in cytochrome c level in cytosol at 50 uM incubated upto 48 hrs by immunoblot analysis
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