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Enzyme Inhibition Assay from Article 10.1016/j.bmc.2006.06.050: "Synthesis and structure activity relationships of novel non-peptidic metallo-aminopeptidase inhibitors."
Assay data:7 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 19 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of aeromonas proteolytica aminopeptidase using L-leucine-p-nitroanilide as substrate by spectrophotometry
Assay data:1 Active, 1 Activity ≤ 1 µM, 4 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Inhibition of Aeromonas proteolytica aminopeptidase assessed as hydrolysis of LeuNA at pH 8 by spectrophotometric analysis
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Inhibition of aeromonas proteolytica aminopeptidase
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of Aeromonas proteolytica leucyl aminopeptidase using L-leucine para-notroanilide as substrate assessed as release of para-nitroaniline by Dixon plot analysis
Assay data:3 Active, 2 Activity ≤ 1 µM, 7 Tested
Inhibition of Aeromonas proteolytica aminopeptidase using L-leucine-p-nitroanilide as substrate after 30 mins by Dixon plot analysis
Assay data:12 Tested
Inhibition of Aeromonas proteolytica aminopeptidase by Dixon plot analysis
Assay data:1 Active, 1 Activity ≤ 1 µM, 9 Tested
Inhibition of metalloprotease from family M28, Aeromonas proteolytica aminopeptidase
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Inhibition of aeromonas proteolytica aminopeptidase at 5 uM incubated at pH 8 and 30 degC followed by addition of 50 uM L-leucine-p-nitroanilide substrate by spectrophotometry
Assay data:2 Active, 2 Tested
SummaryCompounds, ActivePubMed Citation
Inhibition of aeromonas proteolytica aminopeptidase up to 100 uM
Assay data:36 Tested
Drug level in HEPES buffer treated with 200 uM (S)-4-sulfamoylphenyl 3-(2-amino-4-methylpentanamido)propane-1-sulfonate in presence of aeromonas proteolytica aminopeptidase by spectrophotometry
SummaryPubMed Citation
Drug level in HEPES buffer treated with 200 uM (S)-4-(trifluoromethyl)phenyl 3-(2-amino-4-methylpentanamido)propane-1-sulfonate in presence of aeromonas proteolytica aminopeptidase by spectrophotometry
Drug level in HEPES buffer treated with 200 uM (S)-4-chlorophenyl 3-(2-amino-4-methylpentanamido)propane-1-sulfonate in presence of aeromonas proteolytica aminopeptidase by spectrophotometry
Drug level in HEPES buffer treated with 50 uM (S)-2-methylquinolin-8-yl 3-(2-amino-4-methylpentanamido)propane-1-sulfonate in presence of aeromonas proteolytica aminopeptidase by spectrophotometry
Drug metabolism in HEPES buffer assessed as aeromonas proteolytica aminopeptidase-mediated Isothiazolidine 1,1-dioxide formation at 200 uM by spectrophotometry
Assay data:3 Tested
Drug metabolism in HEPES buffer assessed as aeromonas proteolytica aminopeptidase-mediated 4-hydroxybenzenesulfonamide formation at 200 uM by spectrophotometry
Assay data:1 Tested
Drug metabolism in HEPES buffer assessed as aeromonas proteolytica aminopeptidase-mediated 4-(trifluoromethyl)phenol formation at 200 uM by spectrophotometry
Drug metabolism in HEPES buffer assessed as aeromonas proteolytica aminopeptidase-mediated 4-chlorophenol formation at 200 uM by spectrophotometry
Drug metabolism in HEPES buffer assessed as aeromonas proteolytica aminopeptidase-mediated Isothiazolidine 1,1-dioxide formation at 50 uM by spectrophotometry
Drug metabolism in HEPES buffer assessed as aeromonas proteolytica aminopeptidase-mediated 2-methylquinolin-8-ol formation at 50 uM by spectrophotometry
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