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Peptidase, Angiotensin Converting Enzyme Eurofins Panlabs panel
Assay data:1 Tested
SummaryRelated BioAssays by Target
Cardioprotective activity in rabbit model assessed as conductivity relaxation at 30 uM
Summary
Cardioprotective activity in rabbit model assessed as conductivity relaxation at 8 uM
Cardioprotective activity in rabbit model assessed as conductivity relaxation at 5.6 uM
Cardioprotective activity in rabbit model assessed as resistance relaxation at 30 uM
Cardioprotective activity in rabbit model assessed as resistance relaxation at 8 uM
Cardioprotective activity in rabbit model assessed as resistance relaxation at 5.6 uM
Antihypertensive activity in rabbit aorta assessed as vasodilation
Assay data:2 Tested
Antihypertensive activity in po dosed rabbit assessed as decrease in 30mmhg of systolic blood pressure measured after 4 to 6 hrs
Assay data:4 Tested
Binding affinity to AT1 in rabbit aorta
Assay data:7 Active, 24 Activity ≤ 1 µM, 24 Tested
Inhibition of SERCA1a in rabbit Sarcoplasmic reticulum assessed as inhibition constant in presence of [gamma-32P]ATP and calcium ionophore A23187 by by coupled enzyme assay
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Binding affinity to recombinant rabbit FBPase expressed in Escherichia coli assessed as maximal activity
Assay data:1 Active, 1 Tested
Antiplatelet activity against platelet-activating factor induced rabbit platelet assessed as inhibition of platelet aggregation at 2 ng/ml relative to control
Antiplatelet activity against collagen-induced rabbit platelet assessed as inhibition of platelet aggregation at 100 ug/ml relative to control
Assay data:3 Tested
Antiplatelet activity against arachidonate-induced rabbit platelet assessed as inhibition of platelet aggregation at 50 ug/ml relative to control
Antiplatelet activity against arachidonate-induced rabbit platelet assessed as inhibition of platelet aggregation at 100 ug/ml relative to control
Inhibition of superoxide anion radical release in rabbit polymorphonuclear leucocytes
Hemolytic activity in rabbit RBC assessed as hemolysis at 100 uM incubated for 6 hrs by Uv-vis spectrophotometric analysis
Binding affinity to angiotensin-converting enzyme in rabbit lung assessed as inhibition constant
Assay data:2 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 2 Tested
Inhibition of rabbit lung angiotensin-converting enzyme
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