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Invivo agonist activity at GPR120 in C57BL/6 mouse assessed as reduction in glucose AUC levels at 30 mg/kg,po and measured upto 120 mins by OGTT test
Assay data:1 Tested
SummaryRelated BioAssays by Target
Agonist activity at mouse GPR120 by calcium flux assay
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Agonist activity at mouse GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assay relative to control
Assay data:7 Tested
SummaryPubMed CitationRelated BioAssays by Target
Agonist activity at mouse GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assay
Assay data:7 Active, 7 Activity ≤ 1 µM, 7 Tested
Agonist activity at mouse FFA4 receptor
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Agonist activity at mouse FFA4 receptor relative to control
Agonist activity at recombinant mouse GPR120 expressed in HEK293 cells
Agonist activity at mouse GPR120 expressed in CHOK1 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assay
Assay data:10 Active, 9 Activity ≤ 1 µM, 11 Tested
Agonist activity at mouse GPR120 expressed in U2OS cells assessed as induction of beta-arrestin2 recruitment after 90 mins by luminescence assay
Assay data:10 Active, 5 Activity ≤ 1 µM, 11 Tested
Agonist activity at mouse GPR120 assessed as induction of IP1 accumulation
Assay data:4 Active, 3 Activity ≤ 1 µM, 5 Tested
Agonist activity at mouse GPR120 assessed as induction of beta-arrestin recruitment
Assay data:4 Active, 4 Activity ≤ 1 µM, 5 Tested
Agonist activity at mouse GPR120 expressed in human U2OS cells assessed as beta-arrestin recruitment after 90 mins by luminescence assay
Agonist activity at mouse GPR120 expressed in CHOK1 cells assessed as increase in IP1 accumulation after 60 mins by HTRF assay
Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested
Agonist activity at mouse GPR120 expressed in CHOK1 cells measured after 60 mins by IP1-HTRF assay relative to basal level
Assay data:35 Tested
Agonist activity at mouse GPR120 expressed in CHOK1 cells measured after 60 mins by IP1-HTRF assay
Assay data:35 Active, 33 Activity ≤ 1 µM, 37 Tested
Agonist activity mouse FFA1 by by BRET based beta-arrestin-2 interaction assay
Agonist activity mouse FFA4 by by BRET based beta-arrestin-2 interaction assay
Agonist activity mouse FFA1 up to 100 uM by Gq-dependent calcium mobilization assay
Assay data:3 Tested
Agonist activity mouse FFA4 by Gq-dependent calcium mobilization assay
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
Genome-wide siRNA screen of genes regulating the Lipopolysaccharide-induced NF-kappaB and TNF-alpha responses in mouse macrophages_Primary screen NFkB readout
Assay data:762 Active, 16821 Tested
SummaryRelated BioAssays by Same Project
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