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Inhibition of PIM2 (unknown origin)
Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested
SummaryRelated BioAssays by Target
No assay from US Patent US11759530: "TKI permeability enhancers"
Assay data:9 Active, 9 Activity ≤ 1 µM, 11 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Binding affinity to human PIM2
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human PIM2 at 1 uM relative to control
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of PIM-2 (unknown origin) at 1 uM
Inhibition of human PIM-2 at 2 uM by DiscoveryX Kinomescan assay relative to control
PIM2 DiscoveRx kinase panel
Pim-2(h) Kinase panel
Inhibition of PIM2 (unknown origin) at 1 uM
Enzyme Assay from US Patent US11229631: "Thiazolecarboxamides and pyridinecarboxamide compounds useful as Pim kinase inhibitors"
Assay data:95 Active, 95 Activity ≤ 1 µM, 108 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Pim Enzyme Assays from US Patent US11053215: "Heterocyclic compounds useful as Pim kinase inhibitors"
Assay data:168 Active, 168 Activity ≤ 1 µM, 168 Tested
Pim Enzyme Assay from US Patent US10828290: "Thiazolecarboxamides and pyridinecarboxamide compounds useful as pim kinase inhibitors"
Assay data:106 Active, 108 Activity ≤ 1 µM, 108 Tested
Enzyme Assay from US Patent US10517858: "Thiazolecarboxamides and pyridinecarboxamide compounds useful as PIM kinase inhibitors"
Assay data:94 Active, 94 Activity ≤ 1 µM, 107 Tested
In Vitro Caliper Kinase Assay from US Patent US9452998: "Protein kinase C inhibitors and methods of their use"
Assay data:6 Active, 6 Activity ≤ 1 µM, 7 Tested
Kinase Binding Assay from US Patent US9434725: "5-azaindazole compounds and methods of use"
Assay data:199 Active, 156 Activity ≤ 1 nM, 199 Activity ≤ 1 µM, 199 Tested
Homogeneous Time Resolved Fluorescence Assay (HTRF) from US Patent US9394297: "Amides as pim inhibitors"
Assay data:306 Active, 109 Activity ≤ 1 nM, 305 Activity ≤ 1 µM, 306 Tested
Assay data:138 Active, 17 Activity ≤ 1 nM, 139 Activity ≤ 1 µM, 139 Tested
Enzyme Assay from US Patent US9321756: "Azole compounds as PIM inhibitors"
Assay data:290 Active, 15 Activity ≤ 1 nM, 291 Activity ≤ 1 µM, 293 Tested
PIM2 Activity Assay from US Patent US9284298: "Pyrazolyl-pyrimidine derivatives as kinase inhibitors"
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Target
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