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Agonist activity at mouse TRMP8 expressed in HEK293 cells
Assay data:2 Tested
SummaryRelated BioAssays by Target
Agonist activity at mouse TRPM8 expressed in HEK293 cells assessed as increase in calcium influx at 1 uM incubated for 1 min by Fluo-4-AM dye based FLIPR assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Agonist activity at mouse TRPM8 expressed in HEK293 cells assessed as increase in calcium influx at 0.3 to 30 uM incubated for 1 min by Fluo-4-AM dye based FLIPR assay
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Agonist activity at mouse TRPM8 expressed in HEK293 cells assessed as increase in intracellular calcium level at 33 uM measured for 2.5 mins by Fluo-8-AM dye based fluorescence assay
Assay data:4 Tested
Inhibition of mouse TRPM8 expressed in HEK293 cells assessed as decrease in methanol-evoked increase in intracellular calcium level at 22 uM preincubated for 2 mins followed by methanol addition measured for 2.5 mins by Fluo8-AM dye-based fluorescence assay relative to control
Assay data:3 Tested
Antagonist activity at mouse TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced intracellular calcium levels preincubated for 2.5 mins followed by icilin addition by CCD-camera-based FLASH luminometric analysis
Assay data:25 Active, 23 Activity ≤ 1 µM, 28 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antagonist activity at TRPM8 in C57/BL6 mouse cerebellar granule cells assessed as inhibition of KCl-induced voltage dependent calcium entry at 10 uM by fura-2-based assay
Assay data:7 Tested
Agonist activity at mouse TRPM8 expressed in HEK293 cells assessed as increase in calcium flux at 50 uM after 60 mins by Fluo-4 NW dye based fluorometric assay relative to menthol
Antagonist activity at mouse TRPM8 expressed in HEK293 cells assessed as inhibition of menthol mediated calcium flux at 0.5 to 50 preincubated for 60 mins followed by menthol addition by Fluo-4 NW dye based fluorometric assay
Assay data:2 Active, 6 Tested
Antagonist activity at mouse TRPM8 expressed in HEK293 cells assessed as inhibition of menthol mediated calcium flux at 50 preincubated for 60 mins followed by menthol addition by Fluo-4 NW dye based fluorometric assay
Assay data:4 Active, 4 Tested
Agonist activity at mouse TRPM8 expressed in HEK293 cells assessed as increase in calcium flux at 0.5 uM after 60 mins by Fluo-4 NW dye based fluorometric assay
Assay data:2 Active, 2 Tested
Agonist at mouse TRPM8 expressed in HEK293 cells assessed as calcium flux at 0.5 to 50 uM after 60 mins by Fluo-4 NW dye based fluorometric assay
Assay data:6 Tested
Agonist activity at mouse TRPM8 expressed in HEK293 cells assessed as increase in calcium flux at 50 uM after 60 mins by Fluo-4 NW dye based fluorometric assay
Assay data:5 Active, 5 Tested
Agonist activity at mouse TRPM8 expressed in TREx-HEK cells at 300 uM by Fluo-4 AM dye-based Ca2+ imaging assay
Assay data:16 Tested
Genome-wide siRNA screen of genes regulating the Lipopolysaccharide-induced NF-kappaB and TNF-alpha responses in mouse macrophages_Primary screen NFkB readout
Assay data:762 Active, 16821 Tested
SummaryRelated BioAssays by Same Project
Genome-wide siRNA screen of genes regulating the Lipopolysaccharide-induced NF-kappaB and TNF-alpha responses in mouse macrophages_Primary screen TNF readout
Assay data:1106 Active, 16821 Tested
Antagonist activity against mouse TRPM8 expressed in T-REx HEK cells assessed as inhibition of cold-induced increase in intracellular Ca2+ accumulation pre-incubated for 3 mins prior to cold stimulation by Fluo-4 AM dye based fluorescence assay
Assay data:4 Active, 13 Tested
Antagonist activity against mouse TRPM8 expressed in T-REx HEK cells assessed as inhibition of icilin-induced increase in intracellular Ca2+ accumulation pre-incubated for 3 mins prior to icilin stimulation by Fluo-4 AM dye based fluorescence assay
Assay data:5 Active, 3 Activity ≤ 1 µM, 13 Tested
Antagonist activity against mouse TRPM8 expressed in T-REx HEK cells assessed as inhibition of menthol-induced increase in intracellular Ca2+ accumulation pre-incubated for 3 mins prior to menthol stimulation by Fluo-4 AM dye based fluorescence assay
Agonist activity at mouse TRPM8 expressed in T-REx HEK cells assessed as increase in intracellular Ca2+ accumulation by Fluo-4 AM dye based fluorescence assay relative to ionomycin
Assay data:13 Tested
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