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Inhibition of HRI (unknown origin) assessed as fold change
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of HRI (unknown origin)
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
EIF2AK1 DiscoveRx kinase panel
SummaryRelated BioAssays by Target
HRI(h) Kinase panel
KinomeScan assay: inhibition of EIF2AK1
Assay data:108 Tested
HRI(EIK1CGQ1) Takeda global kinase panel
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
HRI(h) Eurofins kinase panel
HRI ProQinase selectivity panel
HRI(h) Eurofins Kinase panel
HRI(h) Millipore kinase panel
Inhibition of HRI (unknown origin) assessed as residual activity measured at 1 uM
Assay data:3 Tested
Inhibition of human EIF2AK1 assessed as percent of control at 2000 nM by KINOMEscan assay relative to control
Inhibition of DNA-tagged human EIF2AK1 assessed as percent of control at 50000 nM by qPCR analysis relative to control
Inhibition of human EIF2AK1 assessed as percent of control at 1000 nM by KINOMEscan assay relative to control
Inhibition of wild-type human partial length EIF2AK1 (Q147 to E603 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control
Inhibition of wild-type human partial length EIF2AK1 (Q147 to E603 residues) expressed in mammalian expression system at 1 uM by Kinomescan method relative to control
Binding affinity to wild-type human partial length EIF2AK1 (Q147 to E603 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control
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