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Drug uptake by rat hepatic OATP1A1 transporters expressed in CHO cells at 1 uM relative to control
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
TP_TRANSPORTER: uptake in Oatp1-expressing CHO-03 cell
Assay data:4 Active, 11 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
TP_TRANSPORTER: inhibition of BSP uptake (BSP: 1 uM, Aldosterone: 100 uM) in Oatp1-expressing HeLa cells
TP_TRANSPORTER: inhibition of E217betaG uptake (E217betaG: 0.1 uM, Tolbutamide: 1000 uM) in Oatp1-expressing LLC-PK1 cells
TP_TRANSPORTER: inhibition of Fexofenadine uptake (Fexofenadine: 1 uM, Apple juice: 5 %) in Oatp1-expressing HeLa cells
TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.01uM, BSP: 250 uM) in Xenopus laevis oocytes
TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.01uM, p-Chlorophenacyl-SG: 1000 uM) in Xenopus laevis oocytes
TP_TRANSPORTER: inhibition of Pravastatin uptake (Pravastatin: 0.5 uM, DHEAS: 50 uM) in Oatp1-expressing 293c18 cells
TP_TRANSPORTER: inhibition of Taurocholate uptake (Taurocholate: 0.5 uM, BMS243887: 50 uM) in Oatp1-expressing 293c18 cells
TP_TRANSPORTER: inhibition of Taurocholate uptake (Taurochorate: 20 uM, GC: 200 uM) in Xenopus laevis oocytes
TP_TRANSPORTER: inhibition of Temocaprilat uptake (Temocaprilat: 0.1 uM, DBSB: 100 uM) in Oatp1-expressing COS-7 cells
TP_TRANSPORTER: uptake in Oatp1-expressing COS-7 cells
TP_TRANSPORTER: uptake in Oatp1-expressing LLC-PK1 cells
Assay data:1 Active, 1 Tested
TP_TRANSPORTER: uptake of Taurolagodeoxycholate at 1 u M in Oatp1-expressing HeLa cells
TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing LLC-PK1 cells
Assay data:1 Active, 3 Tested
TP_TRANSPORTER: uptake in Oatp1-expressing HeLa cells
Assay data:5 Tested
Assay data:3 Active, 6 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
TP_TRANSPORTER: uptake in Xenopus laevis oocytes
Assay data:3 Active, 1 Activity ≤ 1 µM, 6 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Assay data:10 Tested
TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cells
Assay data:11 Active, 15 Tested
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