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Inhibition of p-glycoprotein in docetaxel-resistant human PC-3 cells assessed as inhibition of calcein excretion at 0.39 to 50 uM incubated for 30 mins by fluorescence based plate reader analysis
Assay data:4 Active, 4 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Substrate activity at P-gp (unknown origin) assessed as efflux ratio
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of P-gp in doxorubicin-resistant carbonic anhydrase knockout human A549 cells overexpressing P-gp assessed as Vmax at 3 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Assay data:2 Tested
Inhibition of P-gp in doxorubicin-resistant carbonic anhydrase knockout human A549 cells overexpressing P-gp assessed as Vmax at 1 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant carbonic anhydrase knockout human A549 cells overexpressing P-gp assessed as Km at 3 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of P-gp in doxorubicin-resistant carbonic anhydrase knockout human A549 cells overexpressing P-gp assessed as Km at 1 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant human A549 cells overexpressing P-gp assessed as Vmax at 3 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant human A549 cells overexpressing P-gp assessed as Vmax at 1 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant human A549 cells overexpressing P-gp assessed as Km at 3 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant human A549 cells overexpressing P-gp assessed as Km at 1 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in human A549 cells overexpressing P-gp assessed as Vmax at 3 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in human A549 cells overexpressing P-gp assessed as Vmax at 1 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in human A549 cells overexpressing P-gp assessed as Km at 3 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in human A549 cells overexpressing P-gp assessed as Km at 1 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant carbonic anhydrase knockout human HT-29 cells overexpressing P-gp assessed as Vmax at 3 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant carbonic anhydrase knockout human HT-29 cells overexpressing P-gp assessed as Vmax at 1 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant carbonic anhydrase knockout human HT-29 cells overexpressing P-gp assessed as Km at 3 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant carbonic anhydrase knockout human HT-29 cells overexpressing P-gp assessed as Km at 1 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant human HT-29 cells overexpressing P-gp assessed as Vmax at 3 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
Inhibition of P-gp in doxorubicin-resistant human HT-29 cells overexpressing P-gp assessed as Vmax at 1 uM in presence of 0 to 100 uM doxorubicin measured after 24 hrs
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