BioAssay by Target (List) for Gene (Select 5566) - PubChem BioAssay - NCBI

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Select item 19633221.

Source:: National Center for Advancing Translational Sciences (NCATS)

Deposit Date:: 2024/05/09
Hold-until Date:: 2025/05/09

AID:: 1963322

Select item 19633212.

Source:: National Center for Advancing Translational Sciences (NCATS)

Deposit Date:: 2024/05/09
Hold-until Date:: 2025/05/07

AID:: 1963321

Select item 19624403.

PRKACA Invitrogen Lab (UK) kinase screen (BI)

Source:: ChEMBL

Protein Target:: cAMP-dependent protein kinase catalytic subunit alpha

Assay data:1 Tested

AID:: 1962440

Summary Related BioAssays by Target

Select item 19622934.

PRKACA Invitrogen Lab (UK) kinase screen (BI)

Source:: ChEMBL

Protein Target:: cAMP-dependent protein kinase catalytic subunit alpha

Assay data:1 Tested

AID:: 1962293

Summary Related BioAssays by Target

Select item 19608755.

Inhibition of PKA (unknown origin) at 10 uM by biochemical hotspot kinase assay

Source:: ChEMBL

Protein Targets:: cAMP-dependent protein kinase catalytic subunit alpha; ...
Total:: 3

Assay data:1 Tested

AID:: 1960875

Summary Related BioAssays by Target

Select item 19593606.

Inhibition of PKA (unknown origin) using Kemptide as substrate incubated for [gamma-32P]-ATP incubated for 5 mins by scintillation counter analysis

Source:: ChEMBL

Protein Targets:: cAMP-dependent protein kinase catalytic subunit alpha; ...
Total:: 3

Assay data:1 Active, 1 Tested

AID:: 1959360

Summary Related BioAssays by Target

Select item 19583797.

Inhibition of PKA (unknown origin) at 1 uM relative to control

Source:: ChEMBL

Protein Targets:: cAMP-dependent protein kinase catalytic subunit alpha; ...
Total:: 3

Assay data:3 Tested

AID:: 1958379

Summary Related BioAssays by Target

Select item 19531738.

Inhibition of PKA (unknown origin)

Source:: ChEMBL

Protein Targets:: cAMP-dependent protein kinase catalytic subunit alpha; ...
Total:: 3

Assay data:8 Active, 2 Activity ≤ 1 µM, 11 Tested

AID:: 1953173

Summary Related BioAssays by Target

Select item 19413289.

Inhibition of PKA (unknown origin)

Source:: ChEMBL

Protein Targets:: cAMP-dependent protein kinase catalytic subunit alpha; ...
Total:: 3

Assay data:1 Tested

AID:: 1941328

Summary Related BioAssays by Target

Select item 194106210.

Inhibition of PKA (unknown origin)

Source:: ChEMBL

Protein Targets:: cAMP-dependent protein kinase catalytic subunit alpha; ...
Total:: 3

Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1941062

Summary Related BioAssays by Target

Select item 194105911.

Inhibition of PKA (unknown origin) assessed as fold increase

Source:: ChEMBL

Protein Targets:: cAMP-dependent protein kinase catalytic subunit alpha; ...
Total:: 3

Assay data:1 Tested

AID:: 1941059

Summary Related BioAssays by Target

Select item 193486812.

Inhibition of human recombinant PKA expressed in Escherichia coli at 1 uM by KINOMEscan analysis relative to control

Source:: ChEMBL

Protein Target:: cAMP-dependent protein kinase catalytic subunit alpha

Assay data:1 Tested

AID:: 1934868

Summary Related BioAssays by Target

Select item 193228113.

Inhibition of PKA (unknown origin)

Source:: ChEMBL

Protein Targets:: cAMP-dependent protein kinase catalytic subunit alpha; ...
Total:: 3

Assay data:1 Tested

AID:: 1932281

Summary Related BioAssays by Target

Select item 192187014.

Inhibition of PKA (unknown origin)

Source:: ChEMBL

Protein Targets:: cAMP-dependent protein kinase catalytic subunit alpha; ...
Total:: 3

Assay data:3 Active, 2 Activity ≤ 1 µM, 22 Tested

AID:: 1921870

Summary Related BioAssays by Target

Select item 192086015.

Inhibition of human PKA

Source:: ChEMBL

Protein Targets:: cAMP-dependent protein kinase catalytic subunit gamma; ...
Total:: 3

Assay data:1 Active, 1 Tested

AID:: 1920860

Summary Related BioAssays by Target

Select item 191953516.

In Vitro Kinase Activity Assay from US Patent US11691950: "Isoquinoline-steroid conjugates and uses thereof"

Source:: BindingDB

Protein Targets:: Inhibitor of nuclear factor kappa-B kinase subunit beta; ...
Total:: 16

Assay data:21 Active, 18 Activity ≤ 1 µM, 21 Tested

AID:: 1919535

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191544917.

Selectivity interaction (KinomeScan) EUB0000134b PRKACA

Source:: ChEMBL

Protein Target:: cAMP-dependent protein kinase catalytic subunit alpha

Assay data:1 Tested

AID:: 1915449

Summary Related BioAssays by Target

Select item 191434618.

Selectivity interaction (Enzyme panel (Invitrogen)) EUB0000730a PRKACA

Source:: ChEMBL

Protein Target:: cAMP-dependent protein kinase catalytic subunit alpha

Assay data:1 Active, 1 Tested

AID:: 1914346

Summary Related BioAssays by Target

Select item 191419819.

Selectivity interaction (Kinase panel (University of Dundee)) EUB0000169b PRKACA

Source:: ChEMBL

Protein Target:: cAMP-dependent protein kinase catalytic subunit alpha

Assay data:1 Tested

AID:: 1914198

Summary Related BioAssays by Target

Select item 191413820.

Selectivity interaction (KinomeScan (DiscoverX)) EUB0000716a PRKACA

Source:: ChEMBL

Protein Target:: cAMP-dependent protein kinase catalytic subunit alpha

Assay data:1 Tested

AID:: 1914138

Summary Related BioAssays by Target

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Target

Proteins (8)
BioAssays with protein sequences specified as targets
RNAi Target, Active (8)
BioAssays with gene sequences specified as RNAi targets and the activity is active

BioActivity

Active Compounds (134)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (16)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (101)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Summary (1)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (197)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (41)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose
Chemical Screens (469)
BioAssays reporting BioActivity of chemical reagents
RNAi Screens (44)
BioAssays reporting BioActivity of RNAi reagents
On Hold (2)
On hold BioAssays

Assay Project (4)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (417)
BioAssays extracted from the literature
NIH MLP (9)
BioAssays deposited by the NIH Molecular Libraries Program
Other (88)
BioAssays deposited by other experimentalists

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