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Binding affinity to human activated protein C assessed as inhibition constant using L-Pyroglutamyl-L-prolyl-L-arginine p-Nitroaniline as substrate measured upto 120 mins by spectrophotometric analysis
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition Assay from US Patent US8598206: "Trypsin-like serine protease inhibitors, and their preparation and use"
Assay data:22 Active, 11 Activity ≤ 1 µM, 22 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Serine Protease Inhibition Assay from Article 10.1074/jbc.M409068200: "A selective, slow binding inhibitor of factor VIIa binds to a nonstandard active site conformation and attenuates thrombus formation in vivo."
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human activated protein C using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometry
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of activated Protein C (unknown origin)
Inhibition of human activated Protein C using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysis
Assay data:1 Active, 24 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of human activated protein C preincubated for 15 mins followed by chromogenic substrate addition
Assay data:3 Tested
Inhibition of activated protein C (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate
Assay data:2 Tested
Inhibition of human activated protein C
Inhibition of activated human protein C using pyro-Glu-Pro-Arg-pNA as substrate by spectrophotometry
Inhibition of human activated protein kinase C using H-D-Lys(Cbo)-Pro-Arg-pNA as substrate
Assay data:2 Activity ≤ 1 µM, 2 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of activated protein kinase C (unknown origin)
RNAi screen for vemurafenib enhancer genes in BRAFV600 melanoma - Primary Screen
Assay data:790 Active, 18119 Tested
Summary
Inhibition of human activated protein C using pyro-Glu-Pro-Arg-pNA as substrate at 37 degC after 10 to 120 mins by spectrophotometric method
Inhibition of activated protein C (unknown origin)
Inhibition of human activated protein C by fluorescence based assay
Inhibition of human activated protein C using pyroGlu-Pro-Arg-pNA as substrate after 10 to 120 mins at 37 degC by spectrophotometric method
Assay data:4 Tested
Inhibition of activated protein C (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assay
Human protein C, inactivator of coagulation factors Va and VIIIa (S1: Chymotrypsin)
Assay data:1 Active, 1 Tested
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