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Activation of human 20S proteosome at chymotrypsin like site assessed as maximum fold change in substrate degradation using Suc-LLVY-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by spectrometric analysis relative to control
Assay data:7 Tested
SummaryPubMed CitationRelated BioAssays by Target
Activation of human 20S proteosome at chymotrypsin like site assessed as substrate degradation using Suc-LLVY-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by spectrometric analysis
Assay data:7 Active, 1 Activity ≤ 1 µM, 17 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Activation of human 20S proteosome at trypsin-like site assessed as maximum fold change in substrate degradation using Boc-LLR-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by spectrometric analysis relative to control
Assay data:8 Tested
Activation of human 20S proteosome at trypsin-like site assessed as substrate degradation using Boc-LLR-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by spectrometric analysis
Activation of human 20S proteosome at caspase-like site assessed as maximum fold change in substrate degradation using Z-LLE-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by spectrometric analysis relative to control
Assay data:6 Tested
Activation of human 20S proteosome at caspase-like site assessed as substrate degradation using Z-LLE-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by spectrometric analysis
Assay data:6 Active, 17 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Activation of human 20S proteosome assessed as maximum fold change in substrate degradation using Suc-LLVY-AMC/Z-LLE-AMC/Boc-LLR-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by spectrometric analysis relative to control
Assay data:9 Tested
Activation of human 20S proteosome assessed as substrate degradation using Suc-LLVY-AMC/Z-LLE-AMC/Boc-LLR-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by spectrometric analysis
Inhibition of 20S proteasome subunit beta-5i (unknown origin) using Ac-ANW-AMC as substrate and measured after 30 mins
Assay data:48 Active, 1 Activity ≤ 1 nM, 46 Activity ≤ 1 µM, 50 Tested
Inhibition of chymotrypsin-like activity of 20S proteasome in human MM1.S cells assessed as accumulation of polyubiquitinated proteins at 10 to 1000 nM and measured by Western blot analysis
Assay data:3 Active, 3 Tested
Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-Leu Leu-Val-Tyr-AMC as substrate preincubated for 15 mins followed by substrate addition measured by fluorescence assay
Assay data:25 Active, 1 Activity ≤ 1 nM, 22 Activity ≤ 1 µM, 34 Tested
Inhibition of 20S immunoproteasome beta-5i subunit in human PBMC using Ac-ANW-luciferin substrate preincubated for 2 hrs followed by substrate addition and measured after 30 mins by luminometric analysis
Assay data:36 Active, 33 Activity ≤ 1 µM, 36 Tested
Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and measured after 1 hr by fluorescence intensity assay
Assay data:42 Active, 41 Activity ≤ 1 µM, 42 Tested
Inhibition of human 20S immunoproteasome beta-5i subunit using Ac-ANW-AMC as substrate measured after 1.2 hrs in presence of SDS
Assay data:23 Tested
Inhibition of human proteasome subunit beta type-5i using fluorogenic substrate by UV-spectrometry
Assay data:3 Tested
Inhibition of human 20s proteasome
Assay data:11 Tested
Inhibition of chymotrypsin-like activity of human erythrocytes 20S proteasome using Suc-LLVY-AMC as substrate and measured by fluorescence assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of human 20S proteasome chymotrypsin-like activity at 11 uM using Succ-Leu-Leu-Val-Tyr-AMC as fluorogenic substrate by fluorometric assay
Inhibition of human 20S proteasome caspase-like activity at 11 uM using Cbz-Leu-Leu-Glu-AMC as fluorogenic substrate by fluorometric assay
Inhibition of human 20S proteasome trypsin-like activity at 11 uM using Boc-Leu-Arg-Arg-AMC as fluorogenic substrate by fluorometric assay
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