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Inhibition of human recombinant serine racemase expressed in Escherichia coli Rosetta 2 (DE3) cells using L-serine as substrate by horseradish peroxidase based couple assay
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as reduction in beta-elimination of L-serine at by spectrophotomtery
Assay data:7 Tested
Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as reduction in beta-elimination of L-serine at 330 uM by spectrophotomtery
Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as reduction in beta-elimination of L-serine at 1.2 mM by spectrophotomtery
Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as reduction in beta-elimination of L-serine at 2.8 mM by spectrophotomtery
Assay data:3 Tested
Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as reduction in beta-elimination of L-serine at 5 mM by spectrophotomtery
Assay data:4 Tested
Binding affinity to serine recemase (unknown origin)
Inhibition of full length human recombinant serine recemase C2DC6D mutant expressed in Escherichia coli BL21 (DE3) assessed as D-serine production at 1 mM after 10 mins by Saccharomyces cerevisiae Dsd1SC based D-serine detection assay
Assay data:38 Tested
Inhibition of full length human recombinant serine recemase C2DC6D mutant expressed in Escherichia coli BL21 (DE3) assessed as D-serine production after 10 mins by Saccharomyces cerevisiae Dsd1SC based D-serine detection assay
Assay data:6 Tested
Inhibition of mouse serine racemase by Lineweaver-Burk plot
Assay data:2 Tested
Inhibition of mouse serine racemase using L-serine substrate by reversed-phase HPLC analysis
Assay data:10 Tested
Competitive inhibition of Pseudomonas putida mandelate racemase
Mixed type inhibition of N-terminal 6xHis-tagged recombinant Schizosaccharomyces pombe 972 serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate assessed as enzyme-inhibitor complex preincubated for 2 mins followed by substrate addition by double reciprocal plot analysis
Mixed type inhibition of N-terminal 6xHis-tagged recombinant Schizosaccharomyces pombe 972 serine racemase expressed in Escherichia coli BL21(DE3) using L-serine as substrate assessed as enzyme-substrate-inhibitor complex preincubated for 2 mins followed by substrate addition by double reciprocal plot analysis
Inhibition of N-terminal 6xHis-tagged Clostridium sticklandii ATCC 12662 proline racemase expressed in Escherichia coli BL21(DE3) using L/D-proline as substrate at 142.5 mM preincubated for 5 mins by circular dichroism-based analysis
Inhibition of N-terminal 6xHis-tagged Clostridium sticklandii ATCC 12662 proline racemase expressed in Escherichia coli BL21(DE3) using L/D-proline as substrate preincubated for 5 mins by circular dichroism-based analysis
Noncompetitive inhibition of N-terminal 6xHis-tagged Clostridium sticklandii ATCC 12662 proline racemase expressed in Escherichia coli BL21(DE3) using L/D-proline as substrate preincubated for 5 mins by Cornish-Bowden plot analysis
Competitive inhibition of N-terminal 6xHis-tagged Clostridium sticklandii ATCC 12662 proline racemase expressed in Escherichia coli BL21(DE3) using L/D-proline as substrate
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of Clostridium sticklandii ATCC 12662 proline racemase using L-proline as substrate at 0.36 mM relative to control
Inhibition of Clostridium sticklandii ATCC 12662 proline racemase L-proline as substrate at 57 mM relative to control
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