Related BioAssays, by Target Similarity (List) for PubChem BioAssay (S - PubChem BioAssay - NCBI

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Select item 18017121.

Enzyme Inhibition Assay from US Patent US9156811: "N-myristoyl transferase inhibitors"

Source:: BindingDB

Protein Targets:: Glycylpeptide N-tetradecanoyltransferase; ...
Total:: 2

Assay data:387 Active, 10 Activity ≤ 1 nM, 289 Activity ≤ 1 µM, 505 Tested

AID:: 1801712

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17994802.

Inhibition Assay from Article 10.1016/S1074-5521(02)00240-5: "Crystal structures of Candida albicans N-myristoyltransferase with two distinct inhibitors."

Source:: BindingDB

Protein Targets:: Glycylpeptide N-tetradecanoyltransferase; ...
Total:: 2

Assay data:6 Active, 1 Activity ≤ 1 nM, 5 Activity ≤ 1 µM, 6 Tested

AID:: 1799480

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 16742213.

Inhibition of human NMT1 by fluorescence method

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 3 Tested

AID:: 1674221

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 16527994.

Inhibition of human NMT1 using p60 SRC(2 to 16) as substrate by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:9 Active, 2 Activity ≤ 1 µM, 38 Tested

AID:: 1652799

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 15826635.

Inhibition of human N-myristoyltransferase assessed as reduction in CoASH production by fluorogenic detection based assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 2 Tested

AID:: 1582663

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 15456866.

Inhibition of N-terminal TEV cleavage site-fused His6 tagged human NMT1 (115 to 496 residues) expressed in Escherichia coli rosetta2 cells at 100 uM using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:3 Tested

AID:: 1545686

Summary PubMed Citation Related BioAssays by Target

Select item 15456847.

Inhibition of human NMT1 R295Q/W297F/A452M/L453V/L462V/N473H/L495M/Q496L mutant expressed in Escherichia coli Rosetta-2 cells at 500 uM using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay relative to control

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:3 Tested

AID:: 1545684

Summary PubMed Citation Related BioAssays by Target

Select item 15456838.

Inhibition of N-terminal TEV cleavage site-fused His6 tagged human NMT1 (115 to 496 residues) expressed in Escherichia coli rosetta2 cells at 500 uM using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay relative to control

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:3 Tested

AID:: 1545683

Summary PubMed Citation Related BioAssays by Target

Select item 15456789.

Inhibition of human NMT1 R295Q/N473H/L495M/Q496L mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested

AID:: 1545678

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154567710.

Inhibition of human NMT1 R295Q mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested

AID:: 1545677

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154567611.

Inhibition of human NMT1 W297F/A452M/L453V/L462V/L495M/Q496L mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested

AID:: 1545676

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154567512.

Inhibition of human NMT1 A452M/L453V/L495M mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested

AID:: 1545675

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154567413.

Inhibition of human NMT1 A452M/L453V/L462V mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested

AID:: 1545674

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154567314.

Inhibition of human NMT1 A452M/L453V mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested

AID:: 1545673

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154567215.

Inhibition of human NMT1 L453V mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested

AID:: 1545672

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154567116.

Inhibition of human NMT1 A452M mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested

AID:: 1545671

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154567017.

Inhibition of human NMT1 R295Q/W297F/A452M/L453V/L462V/N473H/L495M/Q496L mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:8 Active, 8 Activity ≤ 1 µM, 8 Tested

AID:: 1545670

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154566918.

Inhibition of human NMT1 Q496L mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:4 Active, 4 Activity ≤ 1 µM, 5 Tested

AID:: 1545669

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154566819.

Inhibition of human NMT1 L495M mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:7 Active, 1 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 8 Tested

AID:: 1545668

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 154566420.

Inhibition of human NMT1 N473H/L495M/Q496L mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after 30 mins by CPM dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Glycylpeptide N-tetradecanoyltransferase 1

Assay data:7 Active, 6 Activity ≤ 1 µM, 8 Tested

AID:: 1545664

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

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Active Compounds (58)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (7)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (53)
BioAssays with the active concentration of tested reagents less than 1 micromolar

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Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

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Literature Extraction (91)
BioAssays extracted from the literature

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