Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
No assay from US Patent US11759530: "TKI permeability enhancers"
Assay data:9 Active, 9 Activity ≤ 1 µM, 11 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Biochemical Assay (10 uM) from US Patent US11685719: "Pyridinone MK2 inhibitors and uses thereof"
Assay data:23 Active, 5 Activity ≤ 1 nM, 24 Activity ≤ 1 µM, 24 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Biochemical Assay (1 uM) from US Patent US11685719: "Pyridinone MK2 inhibitors and uses thereof"
Assay data:23 Active, 2 Activity ≤ 1 µM, 24 Tested
Enzyme-linked immunosorbent assay (ELISA) from US Patent US11655239: "Fused ring pyrimidine amino compound and preparation method, pharmaceutical composition, and use thereof"
Assay data:32 Active, 18 Activity ≤ 1 nM, 32 Activity ≤ 1 µM, 32 Tested
D3R2023 from Article : "Drug Design Data Resource Grand Challenge 3 Dataset: p38a"
Assay data:31 Active, 1 Activity ≤ 1 nM, 22 Activity ≤ 1 µM, 72 Tested
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000304b MAPK14
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (Leadprofiling screen (Ricerca, enzymes, receptors, transporters, and ion channels )) EUB0000347a MAPK14
Selectivity interaction (MSD Pharma/Taiwan screen (enzymes and receptors) ) EUB0000296b MAPK14
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000746a MAPK12
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000263b MAPK12
Selectivity interaction (Kinase panel (University of Dundee)) EUB0000169b MAPK13
Selectivity interaction (Kinase panel (University of Dundee)) EUB0000169b MAPK12
Selectivity interaction (Kinase panel (University of Dundee)) EUB0000169b MAPK11
Selectivity interaction (Kinase panel (University of Dundee)) EUB0000169b MAPK14
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000718a MAPK12
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000713a MAPK14
Selectivity interaction (Western Blot (inhibition of MAPK14 phosphorylation)) EUB0000132b MAPK14
Selectivity interaction (Western Blot (inhibition of HSP27 phosphorylation at Ser82)) EUB0000132b MAPK14
Selectivity interaction (Enzymatic assay) EUB0000624a MAPK14
Affinity Biochemical interaction (ELISA (cell free)) EUB0000718a MAPK14
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on