Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Selectivity interaction (Enzyme panel (Eurofins-Cerep)) EUB0000262b CCKAR
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (CEREP panel (Eurofins, binding assay)) EUB0000262b CCKAR
Agonist activity at human CCK1R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assay
Assay data:7 Active, 3 Activity ≤ 1 nM, 8 Activity ≤ 1 µM, 10 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Cholecystokinin CCK1 (CCKA) Eurofins-Panlabs radioligand binding assay
CCK1 (CCKA) (h) CEREP ligand profiling
CCKA (h) (CCK1) CEREP panel
CCKA/H Eurofins SafetyScreen44 (BI)
CCKAR Eurofins SafetyScan (Receptor)
Radioligand Labeled Binding Assay and Phosphatidylinositol Hydrolysis Assay for the CCK Receptor from Article 10.1021/jm050921q: "Structure-activity relationships of bifunctional peptides based on overlapping pharmacophores at opioid and cholecystokinin receptors."
Assay data:16 Active, 1 Activity ≤ 1 nM, 12 Activity ≤ 1 µM, 16 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
CCK1 (CCKA) (h) Eurofins-Cerep binding assay
Assay data:2 Tested
PRESTO-Tango GPCRome screening (CCKAR)
CCKA (h) (CCK1) CEREP ligand profiling
CCKA/H Cerep selectivity data (BI)
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on