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Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBRET assay
Assay data:26 Active, 25 Activity ≤ 1 µM, 27 Tested
SummaryRelated BioAssays by Target
Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBRET assay
Assay data:26 Active, 22 Activity ≤ 1 µM, 27 Tested
Binding affinity to CK2alpha (unknown origin) assessed as dissociation constant
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of human C-terminal his tagged DYRK1A (26 to 490 residues) expressed in Escherichia coli using DYRKtide (RRRFRPASPLRGPPK) as peptide substrate incubated for 1 hr in presence of ATP by cook activity assay
Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested
Binding affinity to human C-terminal his tagged DYRK1A (26 to 490 residues) expressed in Escherichia coli assessed as apparent dissociation constant
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Binding affinity to human C-terminal his tagged GSK3beta (26 to 383 residues) expressed in Escherichia coli at 12.5 uM by radiometric analysis
Binding affinity to human C-terminal his tagged DYRK1A (26 to 490 residues) expressed in Escherichia coli at 5 uM by radiometric analysis
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Inhibition of human C-terminal his tagged GSK3beta (26 to 383 residues) expressed in Escherichia coli using GYSI(YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE) as peptide substrate incubated for 1 hr in presence of ATP by cook activity assay
Binding affinity to human GSK-3beta assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assay
Assay data:25 Active, 1 Activity ≤ 1 nM, 15 Activity ≤ 1 µM, 37 Tested
Binding affinity to human CLK1 assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assay
Assay data:36 Active, 11 Activity ≤ 1 nM, 37 Activity ≤ 1 µM, 37 Tested
Binding affinity to human DYRK1A assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assay
Assay data:33 Active, 12 Activity ≤ 1 nM, 37 Activity ≤ 1 µM, 37 Tested
Inhibition of recombinant human DYRK1B expressed in Sf9 insect cells using DYRKtide peptide as substrate incubated for 110 mins in presence of ATP by non-radioactive ADP-Glo luminescence microplate reader assay
Assay data:34 Active, 31 Activity ≤ 1 µM, 35 Tested
Inhibition of recombinant human DYRK1A expressed in Escherichia coli using DYRKtide peptide as substrate incubated for 110 mins in presence of ATP by non-radioactive ADP-Glo luminescence microplate reader assay
Assay data:35 Active, 32 Activity ≤ 1 µM, 35 Tested
Inhibition of recombinant human CLK1 expressed in Sf9 insect cells using myelin basic protein as substrate incubated for 110 mins in presence of ATP by non-radioactive ADP-Glo luminescence microplate reader assay
Assay data:32 Active, 29 Activity ≤ 1 µM, 35 Tested
Inhibition of recombinant human DYRK3 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Assay data:28 Active, 13 Activity ≤ 1 µM, 56 Tested
Inhibition of recombinant human DYRK2 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Assay data:37 Active, 20 Activity ≤ 1 µM, 56 Tested
Inhibition of recombinant human DYRK1B expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Assay data:46 Active, 33 Activity ≤ 1 µM, 56 Tested
Inhibition of recombinant human DYRK1A expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Assay data:48 Active, 37 Activity ≤ 1 µM, 56 Tested
Inhibition of recombinant human CLK4 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Assay data:45 Active, 40 Activity ≤ 1 µM, 56 Tested
Inhibition of recombinant human CLK3 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Assay data:31 Active, 11 Activity ≤ 1 µM, 56 Tested
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