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Human gonadotropin-releasing hormone receptor (GnRHR) small molecule agonists, calcium flux assay in GnRHR-HEK293 cells
Assay data:169 Active, 2 Activity ≤ 1 nM, 27 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same Project
Activation of human carbonic anhydrase 1 by stopped flow assay
Assay data:5 Active, 4 Activity ≤ 1 µM, 7 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Agonist activity at human alpha1 beta adrenergic receptor expressed in CHOK1 cells co-expressing Galpha15 assessed as increase in calcium influx by measuring fluorescence intensity by FLIPR assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Agonist activity at human beta1 adrenergic receptor expressed in CHOK1 cells co-expressing Galpha15 assessed as increase in calcium influx by measuring fluorescence intensity by FLIPR assay
Primary qHTS for Huh7 cytotoxicity: counterscreen for inhibitors of MERS-S pseudotyped particle cell entry
Assay data:25 Active, 8 Activity ≤ 1 µM, 2678 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Depositor
Activation of human CA1 by stopped-flow CO2 hydration assay
Assay data:14 Active, 8 Activity ≤ 1 µM, 24 Tested
Acetylcholinesterase (AChE) small molecule antagonists: colormetric cell-based qHTS assay
Assay data:445 Active, 57 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Primary qHTS to identify gynecologic anti-cancer compounds using libraries of approved drugs and bioactive compounds
Assay data:1106 Active, 14 Activity ≤ 1 nM, 6478 Activity ≤ 1 µM, 7578 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Depositor
Activation of Burkholderia pseudomallei gamma carbonic anhydrase at 10 uM incubated for 15 mins prior to testing by stopped flow CO2 hydration assay
Assay data:17 Active, 15 Activity ≤ 1 µM, 19 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Activation of recombinant human carbonic anhydrase 1 at 10 uM incubated for 15 mins prior to testing by stopped flow CO2 hydration assay
Assay data:11 Active, 7 Activity ≤ 1 µM, 19 Tested
Agonist activity at recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane incubated for 30 mins by [35S]GTPgammaS binding assay
Assay data:4 Active, 4 Activity ≤ 1 µM, 17 Tested
Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting method
Assay data:7 Active, 6 Activity ≤ 1 µM, 17 Tested
Displacement of [3H]spiperone from human D2S receptor expressed in CHO cells
Assay data:21 Active, 17 Activity ≤ 1 µM, 25 Tested
Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cells
Assay data:20 Active, 5 Activity ≤ 1 nM, 19 Activity ≤ 1 µM, 25 Tested
Activation of Malassezia globosa beta-carbonic anhydrase incubated for 15 mins prior to testing by stopped flow CO2 hydrase method
Assay data:7 Active, 2 Activity ≤ 1 µM, 19 Tested
qHTS assay to identify small molecule antagonists of the estrogen related receptor signaling pathway with the pleiotropic PPARgamma coactivator (PGC) from Tox21 10K library: Summary
Assay data:462 Active, 149 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS assay to identify small molecule agonists or antagonists of the thyroid stimulating hormone receptor (TSHR) signaling pathway - wild type cell line counter screen: Summary
Assay data:42 Active, 18 Activity ≤ 1 µM, 9667 Tested
Hit Validation Assay to Identify small molecule Aedes aegypti NPYLR7 Agonists [Small Molecule Inhibitors of Mosquito Biting Behavior]
Assay data:28 Active, 54 Activity ≤ 1 µM, 409 Tested
Counter Screen to Identify Specific Small molecule Agonists for Aedes aegypti NPYLR7 Receptor
Assay data:207 Active, 63 Activity ≤ 1 µM, 409 Tested
qHTS assay to identify small molecule agonists or antagonists of the thyroid stimulating hormone receptor (TSHR) signaling pathway - wild type cell line counter screen
Assay data:30 Active, 1 Activity ≤ 1 nM, 15 Activity ≤ 1 µM, 9667 Tested
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