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Inhibition of Bacillus subtilis RuvA/RuvB protein complex helicase activity expressed in Escherichia coli BL21(DE3) assessed as inhibition of HJ branch migration preincubated for 15 mins followed by substrate addition and measured after 1 hr using 5'-FAM labelled 5'-CACTGTGATGCACGATGATTGACGACAGTAGTCAGTGCTGCAGTGGTCAGGTGTC-3' HJ-a duplex DNA as substrate in presence of ATP by PAGE analysis
Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Antibacterial activity against Bacillus subtilis NCIM 2079 assessed as reduction in bacterial growth incubated for 8 hrs by absorbance based assay
Assay data:9 Active, 9 Activity ≤ 1 µM, 9 Tested
Antimicrobial activity against Bacillus subtilis ATCC 23857 assessed as reduction of bacterial growth incubated for 18 hrs by CLSI protocol based broth microdilution method
Assay data:21 Active, 3 Activity ≤ 1 µM, 22 Tested
Antibiotic activity against Bacillus subtilis ATCC6633 assessed as reduction in bacterial cell growth by measuring resazurin reduction incubated for 6 days by fluorescence microplate based assay
Assay data:3 Tested
SummaryPubMed Citation
Antibacterial activity against Bacillus subtilis assessed as inhibition of bacterial growth by microtiter plate method
Assay data:1 Tested
Antibacterial activity against Bacillus subtilis assessed as bacterial growth inhibition by CLSI protocol based broth microdilution assay
Assay data:5 Tested
Inhibition of Bacillus subtilis RuvA/RuvB protein complex helicase activity expressed in Escherichia coli BL21(DE3) assessed as inhibition of HJ branch migration at 50 uM preincubated for 15 mins followed by substrate addition and measured after 1 hr using 5'-FAM labelled 5'-CACTGTGATGCACGATGATTGACGACAGTAGTCAGTGCTGCAGTGGTCAGGTGTC-3' HJ-a duplex DNA as substrate in presence of ATP by PAGE analysis
Antibacterial activity against Bacillus subtilis NCIM 2079 assessed as bacterial growth inhibition incubated for 8 hrs by absorbance based assay
Assay data:9 Tested
Displacement of BODIPY-TR-cadaverine from Bacillus subtilis Lipoteichoic acid at 8 times MIC measured for 30 mins by fluorescence based microplate reader assay relative to control
Displacement of BODIPY-TR-cadaverine from Bacillus subtilis Lipoteichoic acid at 4 times MIC measured for 30 mins by fluorescence based microplate reader assay relative to control
Displacement of BODIPY-TR-cadaverine from Bacillus subtilis Lipoteichoic acid at 2 times MIC measured for 30 mins by fluorescence based microplate reader assay relative to control
Displacement of BODIPY-TR-cadaverine from Bacillus subtilis Lipoteichoic acid at 1 times MIC measured for 30 mins by fluorescence based microplate reader assay relative to control
Induction of drug resistance against Bacillus subtilis CMCC (B) 63501 measured after 16 passages
Assay data:2 Active, 2 Tested
SummaryCompounds, ActivePubMed Citation
Induction of morphological changes in Bacillus subtilis CMCC (B) 63501 assessed as elongation of bacterial cell at 0.5 times MIC for 4 hrs (Rvb = 3 to 5 um) by microscopic analysis
Assay data:4 Tested
Bactericidal activity against Bacillus subtilis CMCC (B) 63501 assessed as inhibition of bacterial growth incubated for 24 hrs by resazurin dye based microtiter plate assay
Antibacterial activity against Bacillus subtilis CMCC (B) 63501 assessed as inhibition of bacterial growth incubated for 20 to 24 hrs by broth micro dilution method
Assay data:24 Tested
Ratio of MBC for bactericidal activity against Bacillus subtilis CMCC (B) 63501 to MIC for antibacterial activity against Bacillus subtilis CMCC (B) 63501
Antibacterial activity against Bacillus subtilis 168 assessed as inhibition of bacterial growth by Muller hinton broth based microdilution assay
Assay data:55 Tested
Disruption of membrane integrity in Bacillus subtilis ATCC 6633 assessed as increase in PI uptake at 16 ug/ml measured after 1 hr by SYTO9/PI staining based fluorometric analysis
Assay data:5 Active, 5 Tested
Disruption of membrane integrity in Bacillus subtilis ATCC 6633 assessed as increase in PI positive cells at 16 ug/ml measured after 1 hr by SYTO9/PI staining based confocal laser scanning microscope analysis
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