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Inhibition of Mycobacterium smegmatis mc2155 menG assessed as inhibition of 2-methyl-3-(3,7,11-trimethyldodeca-2,6,10-trienyl)naphthalene-1,4-dione formation using 2-(3,7,11-trimethyldodeca-2,6,10-trienyl)naphthalene-1,4-dione as substrate incubated for 3 hrs in presence of SAM by HPLC analysis
Assay data:7 Tested
SummaryPubMed Citation
Activation of NDH-2 in Mycobacterium smegmatis MC2 155 inverted membrane vesicles assessed as increase in oxygen consumption rate in presence of NADH by fluorespirometry
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed Citation
Inhibition of DprE1 in Mycolicibacterium smegmatis MC2 155 lysate assessed as reduction in epimerization of P[14C]RPP to DP[14C]A at 70 uM measured after 1.5 hrs in presence of NADH by TLC-based autoradiography
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of DprE1 in Mycolicibacterium smegmatis MC2 155 lysate assessed as reduction in epimerization of P[14C]RPP to DP[14C]A at 700 uM measured after 1.5 hrs in presence of NADH by TLC-based autoradiography
Assay data:4 Active, 6 Tested
Inhibition of STPK in Mycobacterium smegmatis MC2 155 expressing aminoglycoside phophotransferase-8 assessed as growth inhibition at 350 microg/disk after 18 hrs by paper disk method
Assay data:1 Tested
Inhibition of STPK in Mycobacterium smegmatis MC2 155 expressing aminoglycoside phophotransferase-8 assessed as growth inhibition at 25 nmol/disk after 18 hrs in presence of kanamycin by paper disk method
Inhibition of STPK in Mycobacterium smegmatis MC2 155 expressing aminoglycoside phophotransferase-8 assessed as growth inhibition at 5 nmol/disk after 18 hrs in presence of kanamycin by paper disk method
Assay data:3 Tested
Inhibition of STPK in Mycobacterium smegmatis MC2 155 expressing aminoglycoside phophotransferase-8 assessed as growth inhibition at 100 nmol/disk after 18 hrs in presence of kanamycin by paper disk method
Assay data:2 Tested
Inhibition of STPK in Mycobacterium smegmatis MC2 155 expressing aminoglycoside phophotransferase-8 assessed as growth inhibition at 50 nmol/disk after 18 hrs in presence of kanamycin by paper disk method
Assay data:4 Tested
Inhibition of multidrug resistance efflux pump in Mycobacterium smegmatis str. MC2 155 assessed as increase in EtBr accumulation by measuring relative final fluorescence at <= 1/2 times MIC incubated for 60 mins by real-time fluorometry relative to control
Inhibition of multidrug resistance efflux pump in Mycobacterium smegmatis str. MC2 155 assessed as increase in EtBr accumulation by measuring relative final fluorescence at 1/2 times MIC incubated for 60 mins by real-time fluorometry relative to control
Assay data:8 Tested
Inhibition of ATP synathse in Mycobacterium smegmatis str. MC2 155 inverted membrane vesicles assessed as ATP formation pre-incubated for 30 mins before NADH-ADP-phosphate buffer cocktail addition and measured after 60 mins by kinase glow reagent based assay
Assay data:16 Active, 11 Activity ≤ 1 µM, 30 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Inhibition of Mycobacterium smegmatis 155 6His-tagged DNA gyrase B catalytic domain ATPase activity expressed in Escherichia coli BL21 (DE3) pLysS cells assessed as inorganic phosphate release after 120 mins in presence of ATP by malachite green dye based assay
Assay data:15 Active, 1 Activity ≤ 1 µM, 49 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of LfrA in Mycobacterium smegmatis MC2 155 ATCC 700084 assessed as increase in norfloxacin accumulation at 150 ug/ml measured every 5 mins for 35 mins by fluorometric analysis
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of LfrA in Mycobacterium smegmatis MC2 155 ATCC 700084 assessed as increase in norfloxacin accumulation at 12.5 ug/ml measured every 5 mins for 35 mins by fluorometric analysis
Inhibition of LfrA in Mycobacterium smegmatis MC2 155 ATCC 700084 assessed as increase in norfloxacin accumulation at 25 ug/ml measured every 5 mins for 35 mins by fluorometric analysis
Assay data:1 Active, 5 Tested
Inhibition of LfrA in Mycobacterium smegmatis MC2 155 ATCC 700084 assessed as increase in EtBr accumulation at 150 ug/ml measured every 5 mins for 35 mins by fluorometric analysis
Inhibition of LfrA in Mycobacterium smegmatis MC2 155 ATCC 700084 assessed as increase in EtBr accumulation at 12.5 ug/ml measured every 5 mins for 35 mins by fluorometric analysis
Inhibition of LfrA in Mycobacterium smegmatis MC2 155 ATCC 700084 assessed as increase in EtBr accumulation at 50 ug/ml measured every 5 mins for 35 mins by fluorometric analysis
Inhibition of LfrA in Mycobacterium smegmatis MC2 155 ATCC 700084 assessed as increase in EtBr accumulation at 25 ug/ml measured every 5 mins for 35 mins by fluorometric analysis
Assay data:7 Active, 8 Tested
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