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Inhibition of Haemonchus contortus by L4 development assay
Assay data:10 Active, 4 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 10 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Anthelmintic activity against third stage larvae of Haemonchus contortus assessed as inhibition of larval development at 20 uM measured after 7 days by microscopic analysis
Assay data:7 Tested
SummaryPubMed Citation
Anthelmintic activity against third stage larvae of Haemonchus contortus assessed as inhibition of xL3 larval motility at 20 uM measured after 72 hrs
Anti-helmintic activity against fourth stage of Haemonchus contortus larvae assessed as reduction in development of L4 stage incubated for 72 hrs followed by reincubation in humidified environment for 4 days
Assay data:6 Active, 2 Activity ≤ 1 µM, 60 Tested
Anti-helmintic activity against third-stage Haemonchus contortus larvae assessed as inhibition of xL3 motility measured after 72 hrs
Assay data:21 Active, 4 Activity ≤ 1 µM, 60 Tested
Anti-helmintic activity against fourth stage L4 Haemonchus contortus larvae assessed as induction of abnormal morphological phenotype at >= 50 uM after 7 days
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed Citation
Anti-helmintic activity against fourth stage L4 Haemonchus contortus larvae assessed as inhibition of larvae motility at 100 uM after 72 hrs
Assay data:1 Tested
Anti-helmintic activity against third-stage xL3 Haemonchus contortus larvae assessed as inhibition of larvae motility at 100 uM measured after 72 hrs
Assay data:3 Tested
Anti-helmintic activity against third-stage Haemonchus contortus larvae assessed as reduction in development of xL3 stage larvae to L4 stage after 7 days
Anti-helmintic activity against third-stage Haemonchus contortus larvae assessed as reduction in larval motility after 72 hrs
Anti-helmintic activity against fourth stage L4 Haemonchus contortus larvae assessed as induction of changes in internal structure measured on day 7 by light microscopic method
Anti-helmintic activity against fourth stage L4 Haemonchus contortus larvae assessed as induction of eviscerated phenotype measured on day 7 by light microscopic method
Anti-helmintic activity against third-stage Haemonchus contortus larvae assessed as reduction in development of xL3 stage larvae to L4 stage at low concentration after 7 days
Anti-helmintic activity against third-stage Haemonchus contortus larvae assessed as induction of eviscerated phenotype at 100 uM measured on day 7 by light microscopic analysis relative to control
Anti-helmintic activity against third-stage Haemonchus contortus larvae assessed as reduction in development of xL3 stage larvae to L4 stage at 100 uM after 7 days
Assay data:2 Active, 2 Tested
Agonist activity at Heaemonchus contortus UNC-49B/C GABAA receptor expressed in Xenopus laevis oocytes by two-electrode voltage-clamp method
Antihelmintic activity against larval stage of Haemonchus contortus
Assay data:2 Tested
Antihelmintic activity against egg stage of Haemonchus contortus
Antihelmintic activity against Haemonchus contortus L3 larval stage
Nematocidal activity against Haemonchus contortus
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