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Items: 1 to 20 of 67

1.

Practical synthesis of a chromene analog for use as a retinoic acid receptor alpha antagonist lead compound.

Jetson R, Malik N, Luniwal A, Chari V, Ratnam M, Erhardt P.

Eur J Med Chem. 2013 May;63:104-8. doi: 10.1016/j.ejmech.2013.02.012. Epub 2013 Feb 19.

2.

Identification of highly potent retinoic acid receptor alpha-selective antagonists.

Teng M, Duong TT, Johnson AT, Klein ES, Wang L, Khalifa B, Chandraratna RA.

J Med Chem. 1997 Aug 1;40(16):2445-51.

PMID:
9258350
4.

Retinoic acid signaling biomarkers after treatment with retinoic acid and retinoic acid receptor alpha antagonist (Ro 41-5253) in canine testis: an in vitro organ culture study.

Kasimanickam VR, Kasimanickam RK.

Theriogenology. 2013 Jan 1;79(1):10-6. doi: 10.1016/j.theriogenology.2012.09.001. Epub 2012 Oct 25.

PMID:
23102850
5.

A widely used retinoic acid receptor antagonist induces peroxisome proliferator-activated receptor-gamma activity.

Schupp M, Curtin JC, Kim RJ, Billin AN, Lazar MA.

Mol Pharmacol. 2007 May;71(5):1251-7. Epub 2007 Feb 8.

PMID:
17290005
6.

Modulation of Retinoic Acid Receptor Subtypes by 5- and 8-Substituted (Naphthalen-2-yl)-based Arotinoids.

Álvarez S, Lieb M, Martínez C, Khanwalkar H, Rodríguez-Barrios F, Álvarez R, Gronemeyer H, de Lera AR.

ChemMedChem. 2015 Aug;10(8):1378-91. doi: 10.1002/cmdc.201500150. Epub 2015 May 26.

PMID:
26012882
7.

Synthesis and structure-activity relationship of RXR antagonists based on the diazepinylbenzoic acid structure.

Sakaki J, Konishi K, Kishida M, Gunji H, Kanazawa T, Uchiyama H, Fukaya H, Mitani H, Kimura M.

Bioorg Med Chem Lett. 2007 Sep 1;17(17):4808-11. Epub 2007 Jun 30.

PMID:
17651969
9.

Aromatase activity induction in human adipose fibroblasts by retinoic acids via retinoic acid receptor α.

Wilde J, Erdmann M, Mertens M, Eiselt G, Schmidt M.

J Mol Endocrinol. 2013 Sep 10;51(2):247-60. doi: 10.1530/JME-12-0129. Print 2013 Oct.

PMID:
24023268
11.

Role of Ser(289) in RARgamma and its homologous amino acid residue of RARalpha and RARbeta in the binding of retinoic acid.

Zhang ZP, Shukri M, Gambone CJ, Gabriel JL, Soprano KJ, Soprano DR.

Arch Biochem Biophys. 2000 Aug 15;380(2):339-46.

PMID:
10933889
12.
13.

Critical role of the H6-H7 loop in the conformational adaptation of all-trans retinoic acid and synthetic retinoids within the ligand-binding site of RARalpha.

Mailfait S, Thoreau E, Belaiche D, Formstecher And B Sablonniè P.

J Mol Endocrinol. 2000 Jun;24(3):353-64.

PMID:
10828828
15.

Retinoic acid induces neuroblastoma cell death by inhibiting proteasomal degradation of retinoic acid receptor alpha.

Nagai J, Yazawa T, Okudela K, Kigasawa H, Kitamura H, Osaka H.

Cancer Res. 2004 Nov 1;64(21):7910-7.

16.

Involvement of retinoic acid receptor-alpha-mediated signaling pathway in induction of CD38 cell-surface antigen.

Mehta K, McQueen T, Manshouri T, Andreeff M, Collins S, Albitar M.

Blood. 1997 May 15;89(10):3607-14.

PMID:
9160665
18.
19.

Regulation of retinoid-induced differentiation in embryonal carcinoma PCC4.aza1R cells: effects of retinoid-receptor selective ligands.

Mills KJ, Vollberg TM, Nervi C, Grippo JF, Dawson MI, Jetten AM.

Cell Growth Differ. 1996 Mar;7(3):327-37.

20.

The Retinoic Acid Receptor-alpha mediates human T-cell activation and Th2 cytokine and chemokine production.

Dawson HD, Collins G, Pyle R, Key M, Taub DD.

BMC Immunol. 2008 Apr 16;9:16. doi: 10.1186/1471-2172-9-16.

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